Molecule Details
InChIKeyZAGFXXPMKXEROI-UHFFFAOYSA-N
Compound NameN-[2-[4-(4-Cyano-phenoxy)-benzenesulfonyl]-1-(3,4,4-trimethyl-2,5-dioxo-imidazolidin-1-ylmethyl)-ethyl]-N-hydroxy-formamide
Canonical SMILESCN1C(=O)N(CC(CS(=O)(=O)c2ccc(Oc3ccc(C#N)cc3)cc2)N(O)C=O)C(=O)C1(C)C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.8
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.8 pIC50 TTD_MultiTarget
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 8.8 pIC50 TTD_MultiTarget
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.7 IC50 ChEMBL;BindingDB