Molecule Details
InChIKeyZAGCLFXBHOXXEN-JPTLTNPLSA-N
Compound Name(2S,4R)-N-(2-((5-(4-(2,6-Dimethoxy-4-(2-methyl-1-oxo-1,2-dihydro-2,7-naphthyridin-4-yl)benzyl)piperazin-1-yl)pentyl)oxy)-4-(4-methylthiazol-5-yl)benzyl)-1-((S)-2-(1-fluorocyclopropane-1-carboxamido)-3,3-dimethylbutanoyl)-4-hydroxypyrrolidine-2-carboxamide
Canonical SMILESCOc1cc(-c2cn(C)c(=O)c3cnccc23)cc(OC)c1CN1CCN(CCCCCOc2cc(-c3scnc3C)ccc2CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.62
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H8M2 BRD9 Homo sapiens Human PF00439 PF12024 7.9 Kd ChEMBL
P40337 VHL Homo sapiens Human PF01847 PF17211 7.5 Kd ChEMBL
Q15369 ELOC Homo sapiens Human PF03931 7.5 Kd ChEMBL
Q15370 ELOB Homo sapiens Human PF00240 7.5 Kd ChEMBL