Molecule Details
InChIKeyZADYAZTTWZYTSD-UHFFFAOYSA-N
Compound Name5-[1-[(2-chlorophenyl)methyl]-2-[1-[4-(2-methylpropyl)phenyl]ethyl]benzimidazol-5-yl]-3H-1,3,4-oxadiazole-2-thione
Canonical SMILESCC(C)Cc1ccc(C(C)c2nc3cc(-c4n[nH]c(=S)o4)ccc3n2Cc2ccccc2Cl)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P20292 ALOX5AP Homo sapiens Human PF01124 7.3 IC50 ChEMBL;BindingDB
O14684 PTGES Homo sapiens Human PF01124 6.4 IC50 ChEMBL;BindingDB
P09917 ALOX5 Homo sapiens Human PF00305 PF01477 6.2 IC50 ChEMBL;BindingDB