Molecule Details
InChIKeyYZZLLEXNNOPPIX-UHFFFAOYSA-N
Compound Name2-amino-4-(3-hydroxyphenyl)-6-(1H-imidazol-2-ylmethylsulfanyl)pyridine-3,5-dicarbonitrile
Canonical SMILESN#Cc1c(N)nc(SCc2ncc[nH]2)c(C#N)c1-c1cccc(O)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P0DMS8 ADORA3 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB