Molecule Details
InChIKeyYZQBDVJPOXNSJR-ULNSLHSMSA-N
Compound Name(S)-2-((S)-4-((R)-2-acetamido-3-(4-fluorophenyl)propanoyl)-3-(3-guanidinopropyl)-2-oxopiperazin-1-yl)-N-methyl-3-(naphthalen-2-yl)propanamide
Canonical SMILESCNC(=O)[C@H](Cc1ccc2ccccc2c1)N1CCN(C(=O)[C@@H](Cc2ccc(F)cc2)NC(C)=O)[C@@H](CCCN=C(N)N)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
Q01726 MC1R Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB