Molecule Details
InChIKeyYZJYYYWPZRYBLV-UHFFFAOYSA-N
Compound Name5-[2-(Cyclohexylamino)pyridin-4-Yl]-4-Naphthalen-2-Yl-2-(Tetrahydro-2h-Pyran-4-Yl)-2,4-Dihydro-3h-1,2,4-Triazol-3-One
Canonical SMILESO=c1n(C2CCOCC2)nc(-c2ccnc(NC3CCCCC3)c2)n1-c1ccc2ccccc2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.06
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB