Molecule Details
InChIKeyYZJYUACRMOFFJC-UHFFFAOYSA-N
Compound Name[2-Fluoro-4-[[5-fluoro-4-(8-fluoro-4-propan-2-yl-2,3-dihydro-1,4-benzoxazin-6-yl)pyrimidin-2-yl]amino]phenyl]-(4-hydroxypiperidin-1-yl)methanone
Canonical SMILESCC(C)N1CCOc2c(F)cc(-c3nc(Nc4ccc(C(=O)N5CCC(O)CC5)c(F)c4)ncc3F)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 9.3 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 7.5 IC50 ChEMBL;BindingDB