Molecule Details
InChIKeyYZAPRHDGKDEXIQ-UHFFFAOYSA-N
Compound NameN-{2-(Formyl-hydroxy-amino)-3-[4-(4-trifluoromethoxy-phenoxy)-benzenesulfonyl]-propyl}-N-methyl-methanesulfonamide
Canonical SMILESCN(CC(CS(=O)(=O)c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)N(O)C=O)S(C)(=O)=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.34
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.8 IC50 ChEMBL;BindingDB
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 8.3 pIC50 TTD_MultiTarget
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.9 pIC50 TTD_MultiTarget