Molecule Details
InChIKeyYYAWOSLKARYYMV-CQSZACIVSA-N
Compound Name[(3R)-4-(4-chlorobenzyl)-7-fluoro-5-acetyl-1,2,3,4-tetrahydrocyclopenta-[b]indol-3-yl]acetic acid
Canonical SMILESCC(=O)c1cc(F)cc2c3c(n(Cc4ccc(Cl)cc4)c12)[C@@H](CC(=O)O)CC3
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13258 PTGDR Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P21731 TBXA2R Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P43116 PTGER2 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB