Molecule Details
InChIKeyYYABRKAKAPIQDP-UHFFFAOYSA-N
Compound Name8-(6,7-Dimethoxy-isoquinolin-4-ylmethyl)-3-isobutyl-1-methyl-3,7-dihydro-purine-2,6-dione
Canonical SMILESCOc1cc2cncc(Cc3nc4c([nH]3)c(=O)n(C)c(=O)n4CC(C)C)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.03
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O76074 PDE5A Homo sapiens Human PF01590 PF00233 8.1 IC50 ChEMBL;BindingDB
Q13370 PDE3B Homo sapiens Human PF00233 6.5 IC50 ChEMBL
Q14432 PDE3A Homo sapiens Human PF00233 6.5 IC50 ChEMBL