Molecule Details
InChIKeyYXTJOVZVHZIUNM-UHFFFAOYSA-N
Compound Name2-tert-Butyl-4-(4-fluoro-phenyl)-5,6,7,8-tetrahydro-pyrido[4,3-d]pyrimidine
Canonical SMILESCC(C)(C)c1nc2c(c(-c3ccc(F)cc3)n1)CNCC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB