Molecule Details
InChIKeyYXICKOJWVBGVKW-UHFFFAOYSA-N
Compound Name3-[6-(1,4-Diazepan-1-yl)-2-pyridinyl]-5-(6-methylpyrazin-2-yl)-[1,2]thiazolo[5,4-c]pyridine
Canonical SMILESCc1cncc(-c2cc3c(-c4cccc(N5CCCNCC5)n4)nsc3cn2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.2 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 9.0 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.7 Ki ChEMBL;BindingDB