Molecule Details
InChIKeyYWYMUWNXZFMLTG-UHFFFAOYSA-N
Compound Name5-[4-(2-Phenylphenyl)piperazin-1-yl]pyrimidine-2,4-diamine
Canonical SMILESNc1ncc(N2CCN(c3ccccc3-c3ccccc3)CC2)c(N)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.7 IC50 ChEMBL;BindingDB
P07382 Leishmania major Pathogen PF00186 PF00303 8.1 IC50 ChEMBL;BindingDB