Molecule Details
InChIKeyYVZHKKQVYYSSEE-HNNXBMFYSA-N
Compound Name6-[(6S)-1,6-dimethyl-3,6-dihydro-2H-pyridin-4-yl]-8-ethyl-11H-benzo[b][1,4]benzodiazepine
Canonical SMILESCCc1ccc2c(c1)C(C1=C[C@H](C)N(C)CC1)=Nc1ccccc1N2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21728 DRD1 Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.2 IC50 ChEMBL;BindingDB