Molecule Details
InChIKeyYVSQVYZBDXIXCC-UHFFFAOYSA-N
Compound NameTelomestatin
Canonical SMILESCc1oc2nc1-c1nc(co1)-c1nc(co1)-c1nc(co1)-c1nc(co1)-c1nc(co1)C1=NC(CS1)c1nc-2c(C)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.68
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9BX63 BRIP1 Homo sapiens Human PF06733 PF13307 8.7 IC50 BindingDB
O14746 TERT Homo sapiens Human PF12009 PF21399 8.4 IC50 ChEMBL
P27296 dinG Escherichia coli (strain K12) Pathogen PF00270 PF06733 PF13307 8.9 IC50 BindingDB