Molecule Details
InChIKeyYVPYFTVDDPMUSO-UHFFFAOYSA-N
Compound Name4-(6-bromo-13-chloro-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl)-N-[2-(1H-imidazol-5-yl)ethyl]-1-pentanoylpiperazine-2-carboxamide
Canonical SMILESCCCCC(=O)N1CCN(C2c3ccc(Cl)cc3CCc3cc(Br)cnc32)CC1C(=O)NCCc1c[nH]cn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.75
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.9 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.6 IC50 ChEMBL;BindingDB