Molecule Details
InChIKeyYUYSIGQIXVQKCJ-UHFFFAOYSA-N
Compound Name1-{6-[5-(2,6-Difluorophenyl)-1H-indazol-3-yl]pyrazin-2-yl}pyrrolidin-3-amine
Canonical SMILESNC1CCN(c2cncc(-c3n[nH]c4ccc(-c5c(F)cccc5F)cc34)n2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB