Molecule Details
InChIKeyYUJACPUEEGUFHA-UHFFFAOYSA-N
Compound NameN-{1-[2-Amino-6-(3-amino-1H-indazol-6-yl)-4-pyrimidinyl]-3-piperidinyl}benzamide
Canonical SMILESNc1nc(-c2ccc3c(N)n[nH]c3c2)cc(N2CCCC(NC(=O)c3ccccc3)C2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.47
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75716 STK16 Homo sapiens Human PF00069 7.6 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
O15530 PDPK1 Homo sapiens Human PF14593 PF00069 7.2 IC50 ChEMBL;BindingDB