Molecule Details
InChIKeyYUGHQIHRDKJIHS-UHFFFAOYSA-N
Compound Name5,6-Dichloro-1-[6-(2-methylpyridin-3-yloxy)pyridin-3-ylcarbamoyl]indoline
Canonical SMILESCc1ncccc1Oc1ccc(NC(=O)N2CCc3cc(Cl)c(Cl)cc32)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB