Molecule Details
InChIKeyYUGGSPPVYUNNGK-UHFFFAOYSA-N
Compound Name6-[1-[2-(1H-indol-4-yloxy)ethyl]piperidin-4-yl]oxy-4H-1,4-benzoxazin-3-one
Canonical SMILESO=C1COc2ccc(OC3CCN(CCOc4cccc5[nH]ccc45)CC3)cc2N1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.4
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 Clinical TTD_MultiTarget TTD_MultiTarget