Molecule Details
InChIKeyYTJXXDVLDUKYHV-LJAQVGFWSA-N
Compound NameN-[(1r)-1-(3,4'-Difluorobiphenyl-4-Yl)-2-(1h-Imidazol-1-Yl)ethyl]-4-(5-Phenyl-1,3,4-Oxadiazol-2-Yl)benzamide
Canonical SMILESO=C(N[C@@H](Cn1ccnc1)c1ccc(-c2ccc(F)cc2)cc1F)c1ccc(-c2nnc(-c3ccccc3)o2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16850 CYP51A1 Homo sapiens Human PF00067 7.0 Kd ChEMBL;BindingDB
Q7Z1V1 CYP51 Trypanosoma cruzi (strain CL Brener) Pathogen PF00067 8.2 Kd ChEMBL;BindingDB
A2TEF2 Leishmania infantum Pathogen PF00067 8.1 Kd ChEMBL;BindingDB