Molecule Details
InChIKeyYTINZZFBHWSAGL-UHFFFAOYSA-N
Compound Name4-[4-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxymethyl]phenyl]methyl]piperazin-1-yl]-3-fluorobenzonitrile
Canonical SMILESN#Cc1ccc(N2CCN(Cc3ccc(COc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)cc3)CC2)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.01
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25100 ADRA1D Homo sapiens Human PF00001 6.0 IC50 ChEMBL
P35348 ADRA1A Homo sapiens Human PF00001 6.0 IC50 ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 6.0 IC50 ChEMBL