Molecule Details
InChIKeyYTHGWGKRZLUTAJ-UHFFFAOYSA-N
Compound Name1-Ethyl-2-{7-[1-(1-imino-ethyl)-piperidin-4-yloxy]-3-oxo-2,3-dihydro-benzo[1,4]oxazin-4-ylmethyl}-1H-indole-6-carboxamidine
Canonical SMILESCCn1c(CN2C(=O)COc3cc(OC4CCN(C(C)=N)CC4)ccc32)cc2ccc(C(=N)N)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 8.7 IC50 ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.1 IC50 ChEMBL;BindingDB