Molecule Details
InChIKeyYSXVOIJEAUPIBJ-UHFFFAOYSA-N
Compound Name2-[[4-Hydroxy-2-oxo-1-[[4-(trifluoromethyl)-1,3-thiazol-2-yl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
Canonical SMILESO=C(O)CNC(=O)c1c(O)c2c(n(Cc3nc(C(F)(F)F)cs3)c1=O)COC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96KS0 EGLN2 Homo sapiens Human PF13640 8.4 IC50 ChEMBL;BindingDB
Q9GZT9 EGLN1 Homo sapiens Human PF13640 PF01753 8.4 IC50 ChEMBL;BindingDB
Q9H6Z9 EGLN3 Homo sapiens Human PF13640 8.1 IC50 ChEMBL;BindingDB