Molecule Details
InChIKeyYRZWSLXIHSDILJ-UHFFFAOYSA-N
Compound Name1-(6-methoxypyrimidin-4-yl)-8-[(3-methyl-2-pyridinyl)methyl]-3-[4-[4-(1H-pyrazol-5-yl)phenyl]phenyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
Canonical SMILESCOc1cc(N2C(=O)N(c3ccc(-c4ccc(-c5ccn[nH]5)cc4)cc3)C(=O)C23CCN(Cc2ncccc2C)CC3)ncn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9GZT9 EGLN1 Homo sapiens Human PF13640 PF01753 8.3 IC50 ChEMBL;BindingDB
Q96KS0 EGLN2 Homo sapiens Human PF13640 8.2 IC50 ChEMBL;BindingDB
Q9H6Z9 EGLN3 Homo sapiens Human PF13640 6.9 IC50 ChEMBL;BindingDB