Molecule Details
InChIKeyYREPTYNUQVYXCF-CQSZACIVSA-N
Compound Name6,7-dimethoxy-~{N}-[(1~{R})-1-naphthalen-1-ylethyl]quinazolin-4-amine
Canonical SMILESCOc1cc2ncnc(N[C@H](C)c3cccc4ccccc34)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P01116 KRAS Homo sapiens Human PF00071 6.5 IC50 ChEMBL;BindingDB
Q07889 SOS1 Homo sapiens Human PF00617 PF00618 PF00621 PF22697 6.5 IC50 ChEMBL
P00533 EGFR Homo sapiens Human PF00757 PF14843 PF07714 PF01030 PF21314 6.2 IC50 ChEMBL;BindingDB