Molecule Details
InChIKeyYQWVLANNJBATDL-UHFFFAOYSA-N
Compound NameN-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4-ylmethyl)-1,2,3,4-tetrahydroquinolin-3-yl]-(4-fluorobenzenesulfonyl)amino]acetamide
Canonical SMILESCn1cncc1CN1CC(N(CC(=O)NC(C)(C)C)S(=O)(=O)Cc2ccc(F)cc2)Cc2cc(C#N)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.38
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5E175 rhlE Aliivibrio fischeri (strain ATCC 700601 / ES114) Pathogen PF00270 PF00271 7.4 IC50 BindingDB
Q5EI73 Plasmodium falciparum Pathogen PF01239 7.4 IC50 ChEMBL