Molecule Details
InChIKeyYQUMEJDEWPVTIF-YMGYHPDWSA-O
Compound Name(2S)-3-(4-hydroxyphenyl)-N-[(3S)-1-[(4-hydroxyphenyl)methyl]-1-methylpiperidin-1-ium-3-yl]-2-[[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]carbamoylamino]propanamide
Canonical SMILESCc1nc(-c2ccc(NC(=O)N[C@@H](Cc3ccc(O)cc3)C(=O)N[C@H]3CCC[N+](C)(Cc4ccc(O)cc4)C3)cc2)no1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P20309 CHRM3 Homo sapiens Human PF00001 8.7 Kd ChEMBL;BindingDB
P08172 CHRM2 Homo sapiens Human PF00001 8.2 Kd ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 6.9 Kd ChEMBL;BindingDB