Molecule Details
InChIKeyYPXNJMUSTWLKRM-UHFFFAOYSA-N
Compound Name9-cyclopentyl-2-N-ethyl-8-N-(2-fluorophenyl)purine-2,8-diamine
Canonical SMILESCCNc1ncc2nc(Nc3ccccc3F)n(C3CCCC3)c2n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.71
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB