Molecule Details
InChIKeyYPXHRVREWGTCMZ-UXHICEINSA-N
Compound NameN-[(1S,2R)-2-phenylcyclopropyl]-4-[4-(2H-tetrazol-5-yl)phenoxy]piperidine-1-carboxamide
Canonical SMILESO=C(N[C@H]1C[C@@H]1c1ccccc1)N1CCC(Oc2ccc(-c3nn[nH]n3)cc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P34913 EPHX2 Homo sapiens Human PF00561 PF00702 8.5 IC50 ChEMBL;BindingDB
P10632 CYP2C8 Homo sapiens Human PF00067 6.1 IC50 ChEMBL;BindingDB