Molecule Details
InChIKeyYPDVNNOPAKMWBO-UHFFFAOYSA-N
Compound NamePyrazolo[1,5-b]pyridazine deriv. 51
Canonical SMILESCc1ccc2c(-c3ccnc(Nc4cccc(C(F)(F)F)c4)n3)cnn2n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.41
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.3 pIC50 TTD_MultiTarget