Molecule Details
InChIKeyYOZAGBCKIMCHID-UHFFFAOYSA-N
Compound NameN-(2,3-difluorophenyl)-2-[3-[[7-[3-[ethyl(2-hydroxyethyl)amino]propoxy]-6-methoxyquinazolin-4-yl]amino]-1H-pyrazol-5-yl]acetamide
Canonical SMILESCCN(CCO)CCCOc1cc2ncnc(Nc3cc(CC(=O)Nc4cccc(F)c4F)[nH]n3)c2cc1OC
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.74
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.4 pIC50 TTD_MultiTarget