Molecule Details
InChIKeyYOSWFXLZVOUMIC-UHFFFAOYSA-N
Compound NameN-(2-adamantyl)-10-cyano-23-oxo-8-oxa-1,15,17,21-tetrazapentacyclo[19.2.2.13,7.19,13.015,19]heptacosa-3,5,7(27),9,11,13(26),16,18-octaene-4-carboxamide
Canonical SMILESN#Cc1ccc2cc1Oc1ccc(C(=O)NC3C4CC5CC(C4)CC3C5)c(c1)CN1CCN(CC1=O)Cc1cncn1C2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.56
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.7 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.6 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 7.4 IC50 ChEMBL