Molecule Details
InChIKeyYOCROJNDVYFOIL-UHFFFAOYSA-N
Compound NamesPLA2-X inhibitor 31
Canonical SMILESNC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1cccc(CCC(=O)O)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O15496 PLA2G10 Homo sapiens Human PF00068 7.1 IC50 ChEMBL;BindingDB
P14555 PLA2G2A Homo sapiens Human PF00068 6.5 IC50 ChEMBL;BindingDB