Molecule Details
InChIKeyYNARAQPWBNWRIS-UHFFFAOYSA-N
Compound Name3-amino-N-[3-(4-aminopiperidin-1-yl)pyridin-2-yl]-6-[6-morpholin-4-yl-3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamide
Canonical SMILESNc1ncc(-c2nc(N3CCOCC3)ccc2C(F)(F)F)nc1C(=O)Nc1ncccc1N1CCC(N)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.66
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P17252 PRKCA Homo sapiens Human PF00130 PF00168 PF00069 PF00433 9.9 IC50 ChEMBL;BindingDB
Q04759 PRKCQ Homo sapiens Human PF00130 PF21494 PF00069 PF00433 9.4 IC50 ChEMBL;BindingDB
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.6 IC50 ChEMBL