Molecule Details
InChIKeyYNACXPCSBHKFII-UHFFFAOYSA-N
Compound Name1-[3-Methoxy-6-[6-(6-methylpyrazin-2-yl)pyrazolo[4,3-c]pyridin-1-yl]-2-pyridyl]hexahydropyrimidin-2-one
Canonical SMILESCOc1ccc(-n2ncc3cnc(-c4cncc(C)n4)cc32)nc1N1CCCNC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.5 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.3 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.7 Ki ChEMBL;BindingDB