Molecule Details
InChIKeyYMUDLHBKUTXRGL-UHFFFAOYSA-N
Compound Name5-[4-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]triazol-1-yl]pyrazolo[1,5-a]pyridine-3-carbaldehyde
Canonical SMILESO=Cc1cnn2ccc(-n3cc(CCCCN4CCN(c5cccc(Cl)c5Cl)CC4)nn3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB