Molecule Details
InChIKeyYLNKOYUKDZZJOW-UHFFFAOYSA-N
Compound Name2-(cyclopropanecarbonylamino)-N-[5-[[1-[(2-fluorophenyl)methyl]piperidin-4-yl]methoxy]-3-pyridinyl]pyridine-4-carboxamide
Canonical SMILESO=C(Nc1cncc(OCC2CCN(Cc3ccccc3F)CC2)c1)c1ccnc(NC(=O)C2CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P22303 ACHE Homo sapiens Human PF08674 PF00135 8.3 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB