Molecule Details
InChIKeyYLNCBZVZEPUMGA-UHFFFAOYSA-N
Compound Name1-[4-[7-(2,6-dimethyl-4-pyridinyl)-5-methyl-9H-carbazol-3-yl]piperidin-1-yl]-2-methylpropan-2-ol
Canonical SMILESCc1cc(-c2cc(C)c3c(c2)[nH]c2ccc(C4CCN(CC(C)(C)O)CC4)cc23)cc(C)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.99
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NYK1 TLR7 Homo sapiens Human PF13855 PF01582 8.8 IC50 ChEMBL;BindingDB
Q9NR97 TLR8 Homo sapiens Human PF13855 PF01582 7.9 IC50 ChEMBL;BindingDB
Q9NR96 TLR9 Homo sapiens Human PF18837 PF13516 PF13855 PF01582 7.2 IC50 ChEMBL;BindingDB