Molecule Details
InChIKeyYLMSOIIFAYJNMX-UHFFFAOYSA-N
Compound Name5-Isopropyl-pyridine-2-sulfonic acid {2-cyclopropyl-5-(2-methoxy-phenoxy)-6-[3-(toluene-4-sulfonylamino)-propoxy]-pyrimidin-4-yl}-amide
Canonical SMILESCOc1ccccc1Oc1c(NS(=O)(=O)c2ccc(C(C)C)cn2)nc(C2CC2)nc1OCCCNS(=O)(=O)c1ccc(C)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24530 EDNRB Homo sapiens Human PF00001 7.7 IC50 ChEMBL;BindingDB
P25101 EDNRA Homo sapiens Human PF00001 7.1 IC50 ChEMBL;BindingDB