Molecule Details
InChIKeyYLBJFQXCNGOXMS-SFTDATJTSA-N
Compound Name(2S,5S)-N,1-dibenzyl-2,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Canonical SMILESC[C@H]1c2ccccc2N(Cc2ccccc2)[C@@H](C)CN1C(=O)NCc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43497 CACNA1G Homo sapiens Human PF00520 6.5 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 6.3 IC50 ChEMBL;BindingDB
Q9P0X4 CACNA1I Homo sapiens Human PF00520 6.0 IC50 ChEMBL