Molecule Details
InChIKeyYKRWZGXTOYQHJI-OAHLLOKOSA-N
Compound Name(6R)-6-(2-aminoethyl)-2-[3-(tert-butylamino)-2-methylquinoxalin-5-yl]-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
Canonical SMILESCc1nc2cccc(-c3cc4c([nH]3)[C@@H](CCN)NC4=O)c2nc1NC(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.5 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.7 IC50 ChEMBL