Molecule Details
InChIKeyYJXVSXOVOPUKHT-UHFFFAOYSA-N
Compound Name3-(2-amino-1,3-benzothiazol-4-yl)-6-pyridin-2-ylsulfonyl-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNc1nc2c(-c3ccc(S(=O)(=O)c4ccccn4)c(S(N)(=O)=O)c3-c3nnn[nH]3)cccc2s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL10.04
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 10.5 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.9 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.7 IC50 BindingDB