Molecule Details
InChIKeyYJPWCVBJBWSWSU-UHFFFAOYSA-N
Compound Name5-Isobutyl-2,2-dimethyl-N-(2-morpholin-4-ylethyl)-1,2,3,4-tetrahydropyrimido[4',5':4,5]thieno[2,3-c]isoquinolin-8-amine
Canonical SMILESCC(C)Cc1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2c1CCC(C)(C)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27815 PDE4A Homo sapiens Human PF18100 PF00233 8.2 IC50 ChEMBL;BindingDB
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 8.1 IC50 ChEMBL;BindingDB
Q08499 PDE4D Homo sapiens Human PF18100 PF00233 7.4 IC50 ChEMBL;BindingDB