Molecule Details
InChIKeyYJEITIRWMUEULI-WNTFFZHHSA-N
Compound NameBoc-Phe-His-Leu-CF3-Ile-Amp
Canonical SMILESCC[C@H](C)[C@H](NC(=O)C(F)(F)C(=O)C(CC(C)C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)NCc1ccccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.62
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00797 REN Homo sapiens Human PF07966 PF00026 8.9 IC50 ChEMBL;BindingDB
P0DJD9 PGA5 Homo sapiens Human PF07966 PF00026 8.3 IC50 ChEMBL;BindingDB