Molecule Details
InChIKeyYJCZMNIYQABZMT-UHFFFAOYSA-N
Compound Name3-[7-[(2-methoxy-3-pyridinyl)methylamino]-3-methyl-1-propan-2-ylpyrazolo[4,5-b]pyridin-5-yl]-1H-pyridin-2-one
Canonical SMILESCOc1ncccc1CNc1cc(-c2ccc[nH]c2=O)nc2c(C)nn(C(C)C)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01064 PDE1B Homo sapiens Human PF00233 PF08499 7.3 IC50 ChEMBL;BindingDB
P54750 PDE1A Homo sapiens Human PF00233 PF08499 6.5 IC50 ChEMBL;BindingDB
Q14123 PDE1C Homo sapiens Human PF00233 PF08499 6.4 IC50 ChEMBL;BindingDB