Molecule Details
InChIKeyYJBGQSYONUDUCN-UHFFFAOYSA-N
Compound Name5-fluoro-N-[5-(4-methylpiperazin-1-yl)-2-pyridinyl]-4-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)pyrimidin-2-amine
Canonical SMILESCN1CCN(c2ccc(Nc3ncc(F)c(-c4cnn5c4CCCC5)n3)nc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.4 Ki ChEMBL;BindingDB
P30281 CCND3 Homo sapiens Human PF02984 PF00134 7.9 Ki ChEMBL
Q00534 CDK6 Homo sapiens Human PF00069 7.4 Ki ChEMBL;BindingDB