Molecule Details
InChIKeyYJBAGQATRBRFBC-UHFFFAOYSA-N
Compound Name5-((4-(2-(4-tert-Butylphenyl)-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)-1-ethylpyrimidine-2,4(1H,3H)-dione
Canonical SMILESCCn1cc(CN2CCN(c3cccc4[nH]c(-c5ccc(C(C)(C)C)cc5)nc34)CC2)c(=O)[nH]c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30968 GNRHR Homo sapiens Human PF00001 8.8 IC50 ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB