Molecule Details
InChIKeyYHYBBOPOIUAVHY-FIRIVFDPSA-N
Compound Name(R)-N-((R)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-((4,4-dimethyl-2-oxooxazolidin-3-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
Canonical SMILESCC1(C)COC(=O)N1CC1(C2CCCCC2)CCN(C(=O)[C@@H](Cc2ccc(Cl)cc2)NC(=O)[C@H]2Cc3ccccc3CN2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 9.1 IC50 ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 7.1 IC50 ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.6 IC50 ChEMBL;BindingDB