Molecule Details
InChIKeyYGSXHXIKDSYAGK-UHFFFAOYSA-N
Compound NameN-ethyl-4-fluoro-N-[4-[1-[2-oxo-2-(6-oxo-5H-benzo[b][1,4]benzodiazepin-11-yl)ethyl]piperidin-4-yl]butyl]benzamide
Canonical SMILESCCN(CCCCC1CCN(CC(=O)N2c3ccccc3NC(=O)c3ccccc32)CC1)C(=O)c1ccc(F)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08172 CHRM2 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB
P20309 CHRM3 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB